Wilson and Gisvold's Textbook of Organic Medicinal and Pharmaceutical Chemistry

1. Introduction 1; 2. Physicochemical properties in relation to biological action 3; 3. Combinatorial chemistry 43; 4. Metabolic changes of drugs and related organic compounds 65; 5. Prodrugs and drug latentiation 142; 6. Biotechnology and drug discovery 160; 7. Immunobiologicals 197; 8. Anti-infective agents 217; 9. Antimalarials 282; 10. Antibacterial antibiotics 299; 11. Antiviral agents 367; 12. Antineoplastic agents 390; 13. Agents for diagnostic imaging 454; 14. Central nervous system depressants 485; 15. Central nervous system stimulants 510; 16. Adrenergic agents 524; 17. Cholinergic drugs and related agents 548; 18. Diuretics 596; 19. Cardiovascular agents 622; 20. Local anesthetic agents 676; 21. Histamine and antihistaminic agents 696; 22. Analgesic agents 731; 23. Steroids and therapeutically related compounds 767; 24. Prostaglandins, leukotrienes, and other eicosanoids 818; 25. Proteins, enzymes, and peptide hormones 830; 26. Vitamins and related compounds 866; 27. An introduction to the medicinal chemistry of herbs 904; 28. Computational chemistry and computer-assisted drug design 919; Appendix: Calculated log P, log D, and pKa 948.